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Graphical contents list • MISCELLANEOUS PDF (998 K) | |||
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Porphyrin–DNA cross-linking agent hybrids: chemical synthesis and biological studies • SHORT COMMUNICATION Hanping He, Tian Tian, Ping Wang, Lin Wu, Jingjing Xu, Xiang Zhou, Xiaolian Zhang, Xiaoping Cao and Xiaojun Wu SummaryPlus | Full Text + Links | PDF (276 K) | |||
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Discovering selective agonists of endothelial target for acetylcholine (ETA) via diversity-guided pharmacophore simplification and simulation • SHORT COMMUNICATION Rifang Yang, Rusheng Zhao, Dongmei Chen, Limei Shan, Liuhong Yun and Hai Wang SummaryPlus | Full Text + Links | PDF (294 K) | |||
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A novel mixed-ligand antimycobacterial dimeric copper complex of ciprofloxacin and phenanthroline • SHORT COMMUNICATION Dilip Kumar Saha, Uday Sandbhor, K. Shirisha, Subhash Padhye, Dileep Deobagkar, Christopher E. Anson and Annie K. Powell SummaryPlus | Full Text + Links | PDF (647 K) | |||
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A new lead compound for abscisic acid biosynthesis inhibitors targeting 9-cis-epoxycarotenoid dioxygenase • SHORT COMMUNICATION Sun-young Han, Nobutaka Kitahata, Tamio Saito, Masatomo Kobayashi, Kazuo Shinozaki, Shigeo Yoshida and Tadao Asami SummaryPlus | Full Text + Links | PDF (300 K) | |||
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Identification and optimization of novel partial agonists of Neuromedin B receptor using parallel synthesis • SHORT COMMUNICATION Stephen J. Shuttleworth, Mike E. Lizarzaburu, Anne Chai and Peter Coward SummaryPlus | Full Text + Links | PDF (392 K) | |||
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A novel series of potent and selective small molecule inhibitors of the complement component C1s • SHORT COMMUNICATION Nalin L. Subasinghe, Farah Ali, Carl R. Illig, M. Jonathan Rudolph, Scott Klein, Ehab Khalil, Richard M. Soll, Roger F. Bone, John C. Spurlino, Renee L. DesJarlais et al. SummaryPlus | Full Text + Links | PDF (308 K) | |||
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Synthesis and pharmacological evaluation of piperidinoalkanoyl-1,2,3,4-tetrahydroisoquinoline derivatives as novel specific bradycardic agents • SHORT COMMUNICATION Hideki Kubota, Toshihiro Watanabe, Akio Kakefuda, Noriyuki Masuda, Kouichi Wada, Noe Ishii, Shuichi Sakamoto and Shin-ichi Tsukamoto SummaryPlus | Full Text + Links | PDF (260 K) | |||
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N-Isoquinolin-5-yl-N′-aralkyl-urea and -amide antagonists of human vanilloid receptor 1 • SHORT COMMUNICATION Michele C. Jetter, Mark A. Youngman, James J. McNally, Sui-Po Zhang, Adrienne E. Dubin, Nadia Nasser and Scott L. Dax SummaryPlus | Full Text + Links | PDF (263 K) | |||
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Synthesis of 1,7-annulated indoles and their applications in the studies of cyclin dependent kinase inhibitors • SHORT COMMUNICATION Guoxin Zhu, Scott E. Conner, Xun Zhou, Ho-Kit Chan, Chuan Shih, Thomas A. Engler, Rima S. Al-awar, Harold B. Brooks, Scott A. Watkins, Charles D. Spencer et al. SummaryPlus | Full Text + Links | PDF (275 K) | |||
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Interaction with the S1 -pocket of urokinase: 8-heterocycle substituted and 6,8-disubstituted 2-naphthamidine urokinase inhibitors • SHORT COMMUNICATIONMichael D. Wendt, Andrew Geyer, William J. McClellan, Todd W. Rockway, Moshe Weitzberg, Xumiao Zhao, Robert Mantei, Kent Stewart, Vicki Nienaber, Vered Klinghofer and Vincent L. Giranda SummaryPlus | Full Text + Links | PDF (420 K) | |||
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The synthesis and antimicrobial evaluation of a new series of isoxazolinyl oxazolidinones • SHORT COMMUNICATION Michele A. Weidner-Wells, Harvey M. Werblood, Raul Goldschmidt, Karen Bush, Barbara D. Foleno, Jamese J. Hilliard, John Melton, Ellyn Wira and Mark J. Macielag SummaryPlus | Full Text + Links | PDF (258 K) | |||
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Bridgehead-methyl analog of SC-53116 as a 5-HT4 agonist • SHORT COMMUNICATION Daniel P. Becker, Daniel L. Flynn and Clara I. Villamil SummaryPlus | Full Text + Links | PDF (242 K) | |||
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A TOPS-MODE approach to predict adenosine kinase inhibition • SHORT COMMUNICATION Maykel Pérez González and Maria del Carmen Terán Moldes SummaryPlus | Full Text + Links | PDF (243 K) | |||
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Image contrast agents activated by prostate specific antigen (PSA) • SHORT COMMUNICATION Graham B. Jones, Longfei Xie, Ahmed El-Shafey, Curtis F. Crasto, Glenn J. Bubley and Anthony V. D’Amico SummaryPlus | Full Text + Links | PDF (261 K) | |||
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Molecular modeling studies on the active binding site of the blood–brain barrier choline transporter • SHORT COMMUNICATION Werner J. Geldenhuys, Paul R. Lockman, James H. McAfee, Kevin T. Fitzpatrick, Cornelis J. Van der Schyf and David D. Allen SummaryPlus | Full Text + Links | PDF (443 K) | |||
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Structural differences between paroxetine and femoxetine responsible for differential inhibition of Staphylococcus aureus efflux pumps • SHORT COMMUNICATION Peng Wei, Glenn W. Kaatz and Robert J. Kerns SummaryPlus | Full Text + Links | PDF (285 K) | |||
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SAR study of a subtype selective allosteric potentiator of metabotropic glutamate 2 receptor, N-(4-phenoxyphenyl)-N-(3-pyridinylmethyl)ethanesulfonamide • SHORT COMMUNICATION David A. Barda, Zhao-Qing Wang, Thomas C. Britton, Steven S. Henry, G. Erik Jagdmann, Darrell S. Coleman, Michael P. Johnson, Sherri L. Andis and Darryle D. Schoepp SummaryPlus | Full Text + Links | PDF (264 K) | |||
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Conformationally restricted analogs of deoxynegamycin • SHORT COMMUNICATION B. Raju, Sampathkumar Anandan, Shihai Gu, Prudencio Herradura, Hardwin O’Dowd, Bum Kim, Marcela Gomez, Corinne Hackbarth, Charlotte Wu, Wen Wang et al. SummaryPlus | Full Text + Links | PDF (281 K) | |||
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Human ACAT-1 and -2 inhibitory activities of saucerneol B, manassantin A and B isolated from Saururus chinensis • SHORT COMMUNICATION Woo Song Lee, Dae-Woo Lee, Young-Il Baek, So-Jin An, Kyung-Hyun Cho, Yang-Kyu Choi, Hyoung-Chin Kim, Ho-Yong Park, Ki-Hwan Bae and Tae-Sook Jeong SummaryPlus | Full Text + Links | PDF (260 K) | |||
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Synthesis and activity of phosphinic tripeptide inhibitors of cathepsin C • SHORT COMMUNICATION Artur Mucha, Ma SummaryPlus | Full Text + Links | PDF (264 K) | |||
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Lingshuiol, a novel polyhydroxyl compound with strongly cytotoxic activity from the marine dinoflagellate Amphidinium sp. • SHORT COMMUNICATION Xiao-Chun Huang, Di Zhao, Yue-Wei Guo, Hou-Ming Wu, Li-Ping Lin, Zhong-Hua Wang, Jian Ding and Yong-Shui Lin SummaryPlus | Full Text + Links | PDF (305 K) | |||
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Novel nonpeptidic inhibitors of HIV-1 protease obtained via a new multicomponent chemistry strategy • SHORT COMMUNICATION Nasser A. M.Yehia, Walfrido Antuch, Barbara Beck, Sibylle Hess, Vesna Schauer-Vuka SummaryPlus | Full Text + Links | PDF (389 K) | |||
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Synthesis and biological evaluation of novel -carboline derivatives as Tat–TAR interaction inhibitors • SHORT COMMUNICATION Xiaolin Yu, Wei Lin, Jingyun Li and Ming Yang SummaryPlus | Full Text + Links | PDF (285 K) | |||
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Development of an isotope-coded activity-based probe for the quantitative profiling of cysteine proteases • SHORT COMMUNICATION Paul F. van Swieten, Rene Maehr, Adrianus M. C. H. van den Nieuwendijk, Benedikt M. Kessler, Michael Reich, Chung-Sing Wong, Hubert Kalbacher, Michiel A. Leeuwenburgh, Christoph Driessen, Gijsbert A. van der Marel et al. SummaryPlus | Full Text + Links | PDF (492 K) | |||
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2-Alkylsulfanyl estrogen derivatives: synthesis of a novel class of multi-targeted anti-tumour agents • SHORT COMMUNICATION Mathew P. Leese, Simon P. Newman, Atul Purohit, Michael J. Reed and Barry V. L. Potter SummaryPlus | Full Text + Links | PDF (250 K) | |||
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Oxazolidinone: search for highly potent antibacterial • SHORT COMMUNICATION Braj Bhushan Lohray, Vidya Bhushan Lohray, Brijesh Kumar Srivastava, Sunil Gupta, Manish Solanki, Prashant Kapadnis, Vijay Takale and Purvi Pandya SummaryPlus | Full Text + Links | PDF (252 K) | |||
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Synthesis and evaluation of nonpeptide substituted spirobenzazepines as potent vasopressin antagonists • SHORT COMMUNICATION Min Amy Xiang, Robert H. Chen, Keith T. Demarest, Joseph Gunnet, Richard Look, William Hageman, William V. Murray, Donald W. Combs, Philip J. Rybczynski and Mona Patel SummaryPlus | Full Text + Links | PDF (255 K) | |||
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An efficient sequence for the preparation of small secondary amine hydrochloride salts for focused library generation without need for distillation or chromatographic purification • SHORT COMMUNICATION Gene M. Dubowchik, Jodi A. Michne and Dmitry Zuev SummaryPlus | Full Text + Links | PDF (242 K) | |||
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Exploring the possible binding sites at the interface of triosephosphate isomerase dimer as a potential target for anti-tripanosomal drug design • SHORT COMMUNICATION L. Michel Espinoza-Fonseca and José G. Trujillo-Ferrara SummaryPlus | Full Text + Links | PDF (319 K) | |||
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In vitro SAR of (5-(2H)-isoxazolonyl) ureas, potent inhibitors of hormone-sensitive lipase • SHORT COMMUNICATION Derek B. Lowe, Steven Magnuson, Ning Qi, Ann-Marie Campbell, James Cook, Zhenqiu Hong, Ming Wang, Mareli Rodriguez, Furahi Achebe, Harold Kluender et al. SummaryPlus | Full Text + Links | PDF (256 K) | |||
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A new 2-carbamoyl pteridine that inhibits mycobacterial FtsZ • SHORT COMMUNICATION R. C. Reynolds, S. Srivastava, L. J. Ross, W. J. Suling and E. L. White SummaryPlus | Full Text + Links | PDF (258 K) | |||
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Structure-based design, synthesis, and antimicrobial activity of purine derived SAH/MTA nucleosidase inhibitors • SHORT COMMUNICATION Martina E. Tedder, Zhe Nie, Stephen Margosiak, Shaosong Chu, Victoria A. Feher, Robert Almassy, Krzysztof Appelt and Kraig M. Yager SummaryPlus | Full Text + Links | PDF (349 K) | |||
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Synthesis of 3-O-acyl/3-benzylidene/3-hydrazone/3-hydrazine/17-carboxyacryloyl ester derivatives of betulinic acid as anti-angiogenic agents • SHORT COMMUNICATION Rama Mukherjee, Manu Jaggi, Praveen Rajendran, Sanjay K. Srivastava, Mohammad J. A. Siddiqui, Anand Vardhan and Anand C. Burman SummaryPlus | Full Text + Links | PDF (308 K) | |||
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5-Alkyl-2-[(aryl and alkyloxylcarbonylmethyl)thio]-6-(1-naphthylmethyl) pyrimidin-4(3H)-ones as an unique HIV reverse transcriptase inhibitors of S-DABO series • SHORT COMMUNICATION Yanping He, Fener Chen, Guangfu Sun, Yueping Wang, Erik De Clercq, Jan Balzarini and Christophe Pannecouque SummaryPlus | Full Text + Links | PDF (254 K) | |||
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Potential hypotensive agents: synthesis and hypotensive activity of oxime ethers derived from 1-naphthoxepines and related compounds • SHORT COMMUNICATION Vishnu K. Tandon, Manoj Kumar, Anoop K. Awasthi, Hari O. Saxena and Gajendra K. Goswamy SummaryPlus | Full Text + Links | PDF (251 K) | |||
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Design and synthesis of -amino- -hydroxy amide derivatives as inhibitors of MetAP2 and HUVEC growth • SHORT COMMUNICATIONMartin Sendzik, James W. Janc, Ronnel Cabuslay, Lee Honigberg, Richard L. Mackman, Catherine Magill, Neil Squires and Nancy Waldeck SummaryPlus | Full Text + Links | PDF (265 K) | |||
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High-throughput identification of fucosyltransferase inhibitors using carbohydrate microarrays • SHORT COMMUNICATION Marian C. Bryan, Lac V. Lee and Chi-Huey Wong SummaryPlus | Full Text + Links | PDF (594 K) | |||
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Synthesis and structure–activity relationships of 3-substituted 1,4-dihydro-4-oxo-1-(2-thiazolyl)-1,8-naphthyridines as novel antitumor agents • SHORT COMMUNICATION Yasunori Tsuzuki, Kyoji Tomita, Yuji Sato, Shigeki Kashimoto and Katsumi Chiba SummaryPlus | Full Text + Links | PDF (263 K) | |||
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Benzimidazoles as new potent and selective DP antagonists for the treatment of allergic rhinitis • SHORT COMMUNICATION Christian Beaulieu, Zhaoyin Wang, Danielle Denis, Gillian Greig, Sonia Lamontagne, Gary O'Neill, Deborah Slipetz and Jennifer Wang SummaryPlus | Full Text + Links | PDF (276 K) | |||
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First total synthesis of structurally unique flavonoids and their strong anti-inflammatory effect • SHORT COMMUNICATION Takashi Nakatsuka, Yoshiaki Tomimori, Yoshiaki Fukuda and Haruo Nukaya SummaryPlus | Full Text + Links | PDF (332 K) | |||
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Development of Yan-Li Song, Peter P. Roller and Ya-Qiu Long SummaryPlus | Full Text + Links | PDF (281 K) | |||
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New highly active taxoids from 9-dihydrobaccatin-9,10-acetals. Part 5 • SHORT COMMUNICATION Yasuyuki Takeda, Kouichi Uoto, Michio Iwahana, Takeshi Jimbo, Motoko Nagata, Ryo Atsumi, Chiho Ono, Noriko Tanaka, Hirofumi Terasawa and Tsunehiko Soga SummaryPlus | Full Text + Links | PDF (322 K) | |||
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1,7-Annulated indolocarbazoles as cyclin-dependent kinase inhibitors • SHORT COMMUNICATION Rima S. Al-awar, James E. Ray, Kyle A. Hecker, Jianping Huang, Philip P. Waid, Chuan Shih, Harold B. Brooks, Charles D. Spencer, Scott A. Watkins, Bharvin R. Patel et al. SummaryPlus | Full Text + Links | PDF (257 K) | |||
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Critical structural motif for the catalytic inhibition of human topoisomerase II by UK-1 and analogs • SHORT COMMUNICATION Ben B. Wang, Nima Maghami, Vanessa L. Goodlin and Paul J. Smith SummaryPlus | Full Text + Links | PDF (328 K) | |||
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Selective urokinase-type plasminogen activator (uPA) inhibitors. Part 3: 1-Isoquinolinylguanidines • SHORT COMMUNICATION Christopher G. Barber, Roger P. Dickinson and Paul V. Fish SummaryPlus | Full Text + Links | PDF (262 K) | |||
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Synthesis and CB1 receptor activities of novel arachidonyl alcohol derivatives • SHORT COMMUNICATION Teija Parkkari, Juha R. Savinainen, Anu L. Rauhala, Tiina L. Tolonen, Tapio Nevalainen, Jarmo T. Laitinen, Jukka Gynther and Tomi Järvinen SummaryPlus | Full Text + Links | PDF (298 K) | |||
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Potent and selective, sulfamide-based human 3-adrenergic receptor agonists • SHORT COMMUNICATION Robert L. Dow, Ernest S. Paight, Steven R. Schneider, John R. Hadcock, Diane M. Hargrove, Kelly A. Martin, Tristan S. Maurer, Nancy A. Nardone, David A. Tess and Paul DaSilva-Jardine SummaryPlus | Full Text + Links | PDF (274 K) | |||
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3,3′-Oxybis(dimethoxytrityl chloride) (O-DMTCl): synthesis and applications of a novel bifunctional protecting group • SHORT COMMUNICATION Natsuhisa Oka, Yogesh S. Sanghvi and Emmanuel A. Theodorakis SummaryPlus | Full Text + Links | PDF (282 K) | |||
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3-(7-Azaindolyl)-4-arylmaleimides as potent, selective inhibitors of glycogen synthase kinase-3 • SHORT COMMUNICATION Han-Cheng Zhang, Hong Ye, Bruce R. Conway, Claudia K. Derian, Michael F. Addo, Gee-Hong Kuo, Leonard R. Hecker, Diane R. Croll, Jian Li, Lori Westover et al. SummaryPlus | Full Text + Links | PDF (330 K) | |||
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Novel thrombin inhibitors incorporating weakly basic heterobicyclic P1-arginine mimetics: optimization via modification of P1 and P3 moieties • SHORT COMMUNICATION Andreja Kranjc, Lucija Peterlin-Ma SummaryPlus | Full Text + Links | PDF (281 K) | |||
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The monoethyl ester of meconic acid is an active site inhibitor of HCV NS5B RNA-dependent RNA polymerase • SHORT COMMUNICATION Paola Pace, Emanuela Nizi, Barbara Pacini, Silvia Pesci, Victor Matassa, Raffaele De Francesco, Sergio Altamura and Vincenzo Summa SummaryPlus | Full Text + Links | PDF (372 K) | |||
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A novel 18-glycyrrhetinic acid analogue as a potent and selective inhibitor of 11-hydroxysteroid dehydrogenase 2 • SHORT COMMUNICATION Nigel Vicker, Xiangdong Su, Harshani Lawrence, Adrian Cruttenden, Atul Purohit, Michael J. Reed and Barry V. L. Potter SummaryPlus | Full Text + Links | PDF (272 K) | |||
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2,3-Dihydro-1,3-dioxo-1H-isoindole-5-carboxylic acid derivatives: a novel class of small molecule heparanase inhibitors • SHORT COMMUNICATION Stephen M. Courtney, Philip A. Hay, Richard T. Buck, Claire S. Colville, David W. Porter, David I. C. Scopes, Faye C. Pollard, Martin J. Page, James M. Bennett, Margaret L. Hircock et al. SummaryPlus | Full Text + Links | PDF (267 K) | |||
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Long chain amines and long chain ammonium salts as novel inhibitors of dynamin GTPase activity • SHORT COMMUNICATION Timothy A. Hill, Luke R. Odell, Annie Quan, Ruben Abagyan, Gemma Ferguson, Phillip J. Robinson and Adam McCluskey SummaryPlus | Full Text + Links | PDF (259 K) | |||
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Simple and an efficient method for the synthesis of 1-[2-dimethylamino-1-(4-methoxy-phenyl)-ethyl]-cyclohexanol hydrochloride: (±) venlafaxine racemic mixtures • SHORT COMMUNICATION Basappa, C. V. Kavitha and K. S. Rangappa SummaryPlus | Full Text + Links | PDF (240 K) | |||
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Carbonic anhydrase inhibitors: the first QSAR study on inhibition of tumor-associated isoenzyme IX with aromatic and heterocyclic sulfonamides • SHORT COMMUNICATION Mona Jaiswal, Padmakar V. Khadikar, Andrea Scozzafava and Claudiu T. Supuran SummaryPlus | Full Text + Links | PDF (361 K) | |||
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Design and synthesis of dysidiolide analogs from vitamin D3: novel class of Cdc25A inhibitors • SHORT COMMUNICATION Rumiko Shimazawa, Toshiyuki Suzuki, Kosuke Dodo and Ryuichi Shirai SummaryPlus | Full Text + Links | PDF (262 K) | |||
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The effect of 6-substituted-4′,4″-difluorobenztropines on monoamine transporters and the muscarinic M1 receptor • SHORT COMMUNICATION Peter Grundt, Theresa A. Kopajtic, Jonathan L. Katz and Amy Hauck Newman SummaryPlus | Full Text + Links | PDF (273 K) | |||
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Novel inhibitors of bacterial protein synthesis: structure–activity relationships for 1,8-naphthyridine derivatives incorporating position 3 and 4 variants • SHORT COMMUNICATION Richard F. Clark, Sanyi Wang, Zhenkun Ma, Moshe Weitzberg, Christopher Motter, Michael Tufano, Rolf Wagner, Yu-Gui Gu, Peter J. Dandliker, Claude G. Lerner et al. SummaryPlus | Full Text + Links | PDF (258 K) | |||
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New substituted triaza-benzo[cd]azulen-9-ones as promising phosphodiesterase-4 inhibitors • SHORT COMMUNICATION Ingrid Devillers, Isabelle Pevet, Henry Jacobelli, Corinne Durand, Véronique Fasquelle, Jocelyne Puaud, Bernard Gaudillière, Moulay Idrissi, François Moreau and Roger Wrigglesworth SummaryPlus | Full Text + Links | PDF (259 K) | |||
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Comparison of inhibitory activity of isomeric triazolopyridine derivatives towards adenosine receptor subtypes or do similar structures reveal similar bioactivities? • SHORT COMMUNICATION Wolfgang Guba, Matthias Nettekoven, Bernd Püllmann, Claus Riemer and Sébastien Schmitt SummaryPlus | Full Text + Links | PDF (350 K) | |||
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Thiol-based SAHA analogues as potent histone deacetylase inhibitors • SHORT COMMUNICATION Takayoshi Suzuki, Akiyasu Kouketsu, Azusa Matsuura, Arihiro Kohara, Shin-ichi Ninomiya, Kohfuku Kohda and Naoki Miyata SummaryPlus | Full Text + Links | PDF (273 K) | |||
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The first synthesis of glucosylgalactosyl hydroxylysine (Glu-Gal-Hyl) an important biological indicator of collagen turnover • SHORT COMMUNICATION Pietro Allevi, Mario Anastasia, Rita Paroni and Andrea Ragusa SummaryPlus | Full Text + Links | PDF (267 K) | |||
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Synthesis of analogues of a potent antitumor saponin OSW-1 • SHORT COMMUNICATION Jacek W. Morzycki, Agnieszka Wojtkielewicz and S SummaryPlus | Full Text + Links | PDF (277 K) | |||
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Carbonic anhydrase inhibitors. Inhibition of the zinc and cobalt  -class enzyme from the archaeon Methanosarcina thermophila with anions • SHORT COMMUNICATIONAlessio Innocenti, Sabrina Zimmerman, James G. Ferry, Andrea Scozzafava and Claudiu T. Supuran SummaryPlus | Full Text + Links | PDF (264 K) | |||
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Nucleosides and nucleotides. Part 226: Alternate-strand triple-helix formation by 3′-3′-linked oligodeoxynucleotides composed of asymmetrical sequences • SHORT COMMUNICATION Shuichi Hoshika, Yoshihito Ueno, Hiroyuki Kamiya and Akira Matsuda SummaryPlus | Full Text + Links | PDF (335 K) | |||
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Preparation of alkylation agents for bulged DNA microenvironments • SHORT COMMUNICATION Farid S. Fouad, Zhen Xi, Irving H. Goldberg and Graham B. Jones SummaryPlus | Full Text + Links | PDF (267 K) | |||
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Anti-AIDS agents. Part 58: Synthesis and anti-HIV activity of 1-thia-di-O-(−)-camphanoyl-(+)-cis-khellactone (1-thia-DCK) analogues • SHORT COMMUNICATION Peng Xia, Zhi-Jian Yin, Ying Chen, Qian Zhang, Beina Zhang, Yi Xia, Zheng-Yu Yang, Nicole Kilgore, Carl Wild, Susan L. Morris-Natschke and Kuo-Hsiung Lee SummaryPlus | Full Text + Links | PDF (255 K) | |||
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N2-Benzyl-N1-(1-(1-naphthyl)ethyl)-3-phenylpropane-1,2-diamines and conformationally restrained indole analogues: development of calindol as a new calcimimetic acting at the calcium sensing receptor • SHORT COMMUNICATION Albane Kessler, Hélène Faure, Christophe Petrel, Martial Ruat, Philippe Dauban and Robert H. Dodd SummaryPlus | Full Text + Links | PDF (289 K) | |||
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Potent S1P receptor agonists replicate the pharmacologic actions of the novel immune modulator FTY720 • SHORT COMMUNICATION Jeffrey J. Hale, William Neway, Sander G. Mills, Richard Hajdu, Carol Ann Keohane, Mark Rosenbach, James Milligan, Gan-Ju Shei, Gary Chrebet, James Bergstrom et al. SummaryPlus | Full Text + Links | PDF (284 K) | |||
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A new approach to the synthesis of optically active alkylated adenine derivatives • SHORT COMMUNICATION N. F. Zakirova, A. V. Shipitsyn, E. F. Belanov and M. V. Jasko SummaryPlus | Full Text + Links | PDF (264 K) | |||
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Corrigendum to "Hydroxytriamides as potent -secretase inhibitors": [Bioorg. Med. Chem. Lett. 14 (2004) 1917] • ERRATUM C. V. C. Prasad, Owen B. Wallace, Jeffrey W. Noonan, Charles P. Sloan, Wai Lau, Shikha Vig, Michael F. Parker, David W. Smith, Steven B. Hansel, Craig T. Polson et al. SummaryPlus | Full Text + Links | PDF (204 K) | |||
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Corrigendum to "Bridged bicyclic vasopressin receptor antagonists with V2-selective or dual V1a/V2 activity": [Bioorg. Med. Chem. Lett. 12 (2002) 3081] • ERRATUM Alexey B. Dyatkin, William J. Hoekstra, Dennis J. Hlasta, Patricia Andrade-Gordon, Lawrence de Garavilla, Keith T. Demarest, Joseph W. Gunnet, William Hageman, Richard Look and Bruce E. Maryanoff SummaryPlus | Full Text + Links | PDF (207 K) | |||
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Editorial board • MISCELLANEOUS PDF (198 K) | |||
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Contributors to this issue • MISCELLANEOUS PDF (197 K) | |||
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Instructions to contributors • PUBLISHER'S NOTE PDF (74 K) | |||
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